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CTEP (RO4956371)

Manufacturer: ApexBio
Shipping: Standard

Description : CTEP (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM.

Targets : mGlu5 receptor

IC50 : 2.2 nM

Chemical Properties

Cas No. : 871362-31-1

SDF : Download SDF

Chemical Name : 2-chloro-4-[2-[2,5-dimethyl-1-[4-(trifluoromethoxy)phenyl]imidazol-4-yl]ethynyl]pyridine

Canonical SMILES : CC1=C(N=C(N1C2=CC=C(C=C2)OC(F)(F)F)C)C#CC3=CC(=NC=C3)Cl

Formula : C19H13ClF3N3O

M.Wt : 391.77

Solubility : Soluble in DMSO > 10 mM

Storage : Store at -20°C

General tips  : For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.

Shipping Condition : Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request

SizeCatalogue noPrice 
5mg size B1633 £124.00/€173.60
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10mg size B1633-10 £190.00/€266.00
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25mg size B1633-25 £380.00/€532.00
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50mg size B1633-50 £732.00/€1,024.80
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All prices shown are exlusive of VAT.